Publikationen - Institut für Radiopharmazeutische Krebsforschung - Jahr 2014
15 Publikationen2014
Internal Dose Assessment of (-)-18F-Flubatine, Comparing Animal Model Datasets of Mice and Piglets with First-in-Human Results
Sattler, B.; Kranz, M.; Starke, A.; Wilke, S.; Donat, C. K.; et al. (15 authors)
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Journal of Nuclear Medicine 55(2014)11, 1885-1892
DOI: 10.2967/jnumed.114.137059
ISSN: 2159-662X
Synthesis and evaluation of a 18F-labeled spirocyclic piperidine derivative as promising σ1 receptor imaging agent
Chen, Y.-Y.; Wang, X.; Zhang, J.-M.; Deuther-Conrad, W.; Zhang, X.-J.; et al. (12 authors)
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Bioorganic & Medicinal Chemistry 22(2014), 5270-5278
DOI: 10.1016/j.bmc.2014.08.003
Novel Cyclopentadienyl Tricarbonyl 99mTc Complexes Containing 1‑Piperonylpiperazine Moiety: Potential Imaging Probes for Sigma‑1 Receptors
Wang, X.; Li, D.; Deuther-Conrad, W.; Lu, J.; Xie, Y.; et al. (11 authors)
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Journal of Medicinal Chemistry 57(2014), 7113-7125
DOI: 10.1021/jm5009488
Adenosine activates brown adipose tissue and recruits beige adipocytes via A2A receptors
Gnad, T.; Scheibler, S.; von Kügelgen, I.; Scheele, C.; Kilic, A.; et al. (21 authors)
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Nature 516(2014), 395-399
DOI: 10.1038/nature13816
Evaluation of metabolism, plasma protein binding and other biological parameters after administration of (−)-[18 F]Flubatine in humans
Patt, M.; Becker, G. A.; Grossmann, U.; Habermann, B.; Schildan, A.; et al. (17 authors)
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Nuclear Medicine and Biology 41(2014), 489-494
DOI: 10.1016/j.nucmedbio.2014.03.018
Imaging of α7 nicotinic acetylcholine receptors in brain and cerebral vasculature of juvenile pigs with [18F]NS14490
Rötering, S.; Deuther-Conrad, W.; Cumming, P.; Donat, C. K.; Scheunemann, M.; et al. (12 authors)
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EJNMMI Research 4(2014), 1-11
DOI: 10.1186/s13550-014-0043-5
Early increase of cannabinoid receptor density after experimental traumatic brain injury in the newborn piglet
Donat, C. K.; Fischer, F.; Walter, B.; Deuther-Conrad, W.; Brodhun, M.; et al. (7 authors)
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Acta Neurobiologiae Experimentalis 74(2014), 197-210
ISSN: 0365-0820
Distinctive In Vivo Kinetics of the New Sigma1 Receptor Ligands (R)-(+) and (S)-(-)- 18F-Fluspidine in Porcine Brain
Brust, P.; Deuther-Conrad, W.; Becker, G.; Patt, M.; Dont, C. K.; et al. (15 authors)
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Journal of Nuclear Medicine 55(2014)10, 1730-1736
DOI: 10.2967/jnumed.114.137562
ISSN: 0161-5505
Asymmetric Synthesis of Spirocyclic 2-Benzopyrans for Positron Emission Tomography of σ1 Receptors in the Brain
Holl, K.; Schepmann, D.; Fischer, S.; Ludwig, F. A.; Hiller, A.; et al. (9 authors)
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Pharmaceuticals 7(2014), 78-112
DOI: 10.3390/ph7010078
ISSN: 1424-8247
Synthesis and biological evaluation of both enantiomers of [18F]flubatine, promising radiotracers with fas kinetics for the imaging of α4β2-nicotinic acetylcholine receptors
Smits, R.; Fischer, S.; Hiller, A.; Deuther-Conrad, W.; Wenzel, B.; et al. (11 authors)
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Bioorganic & Medicinal Chemistry 22(2014), 804-812
DOI: 10.1016/j.bmc.2013.12.011
Development of 18F-labeled radiotracers for neuroreceptor imaging with positron emission tomography
Brust, P.; van den Hoff, J.; Steinbach, J.
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Neuroscience Bulletin 30(2014)5, 777-811
DOI: 10.1007/s12264-014-1460-6
ISSN: 1995-8218
Hydroxyalkylation with Cyclic Sulfates: Synthesis of Carbazole Derived CB2 Ligands with Increased Polarity
Lueg, C.; Galla, F.; Frehland, B.; Schepmann, D.; Daniliuc, C. G.; et al. (8 authors)
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Archiv der Pharmazie 347(2014), 21-31
DOI: 10.1002/ardp.201300255
Automation of the radiosynthesis and purification procedures for [18F]Fluspidine preparation, a new radiotracer for clinical investigations in PET imaging of σ1 receptors in brain.
Maisonial-Besset, A.; Funke, U.; Wenzel, B.; Fischer, S.; Holl, K.; et al. (8 authors)
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Applied Radiation and Isotopes 84(2014), 1-7
DOI: 10.1016/j.apradiso.2013.10.015
Molecular Imaging of σ1 Receptors In Vivo: Current Status and Perspectives
Brust, P.; Deuther-Conrad, W.; Lehmkuhl, K.; Jia, H.; Wünsch, B.
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Current Medicinal Chemistry 21(2014)1, 35-69
DOI: 10.2174/09298673113209990214
Fluorine containing 6,7-dialkoxybiaryl-based inhibitors for phosphodiesterase 10A: Synthesis and in vitro evaluation of inhibition potency, selectivity and metabolism
Schwan, G.; Asskar, G. B.; Höfgen, N.; Kubicova, L.; Funke, U.; et al. (12 authors)
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ChemMedChem 9(2014)7, 1476-1487
DOI: 10.1002/cmdc.201300522
ISSN: 1860-7187
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