Publications of Institute of Radiopharmaceutical Cancer Research
1325 Publications2012
Irradiation affects cellular properties and Eph receptor expression in human melanoma cells
Mosch, B.; Pietzsch, D.; Pietzsch, J.
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Cell Adhesion & Migration 6(2012)2, 113-125
DOI: 10.4161/cam.20655
ISSN: 1933-6918
A method for model-free partial volume correction in oncological PET
Hofheinz, F.; Langner, J.; Petr, J.; Beuthien-Baumann, B.; Oehme, L.; et al. (8 authors)
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EJNMMI Research 2(2012)16
DOI: 10.1186/2191-219X-2-16
ISSN: 2191-219X
Radioiodinated sunitinib as a potential radiotracer for imaging angiogenesis - radiosynthesis and first radiopharmacological evaluation of 5-[125I]Iodo-sunitinib
Kuchar, M.; Oliveira, M. C.; Gano, L.; Santos, I.; Knieß, T.
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Bioorganic & Medicinal Chemistry Letters 22(2012), 2850-2855
DOI: 10.1016/j.bmcl.2012.02.068
Radiohalogenated 4-anilinoquinazoline-based EGFR-TK inhibitors as potential cancer imaging agents
Neto, C.; Fernandes, C.; Oliveira, M. C.; Gano, L.; Mendes, F.; et al. (7 authors)
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Nuclear Medicine and Biology 39(2012), 247-260
DOI: 10.1016/j.nucmedbio.2011.09.001
Ecto-ATPase inhibition: ATP and adenosine release under physiological and ischemic in vivo conditions in the rat striatum
Melani, A.; Corti, F.; Stephan, H.; Müller, C. E.; Donati, C.; et al. (8 authors)
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Experimental Neurology 233(2012), 193-204
DOI: 10.1016/j.expneurol.2011.09.036
Study of differences in the VEGFR2 inhibitory activities between semaxanib and SU5205 using 3D-QSAR, docking, and molecular dynamics simulations
Munoza, C.; Adasmea, F.; Alzate-Morales, J. H.; Vergara-Jaquea, A.; Kniess, T.; et al. (6 authors)
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Journal of Molecular Graphics and Modelling 32(2012), 39-48
DOI: 10.1016/j.jmgm.2011.10.005
Radiolabeled small molecule inhibitors of VEGFR – recent advances
Kniess, T.
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Current Pharmaceutical Design 18(2012), 2867-2874
DOI: 10.2174/138161212800672796
ISSN: 1873-4286
Module-assisted preparation of 64Cu with high specific activity
Thieme, S.; Walther, M.; Pietzsch, H.-J.; Henniger, J.; Preusche, S.; et al. (7 authors)
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Applied Radiation and Isotopes 70(2012), 602-608
DOI: 10.1016/j.apradiso.2012.01.019
SUV-measurements and patient-specific corrections thereof in pediatric Hodgkin-lymphoma: Is there a benefit for PPV in early response assessment by FDG-PET?
Furth, C.; Meseck, R. M.; Steffen, I. G.; Schoenberger, S.; Denecke, T.; et al. (12 authors)
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Pediatric Blood & Cancer 59(2012), 475-480
DOI: 10.1002/pbc.24047
Automatic volume delineation in oncological PET. Evaluation of a dedicated software tool and comparison with manual delineation in clinical data sets
Hofheinz, F.; Pötzsch, C.; Oehme, L.; Beuthien-Baumann, B.; Steinbach, J.; et al. (7 authors)
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Nuklearmedizin 51(2012), 9-16
DOI: 10.3413/Nukmed-0419-11-07
ISSN: 0029-5566
Synthesis and Molecular Structure of tert-Butyl 4-(2-tert-butoxy-2-oxoethyl)piperazine-1-carboxylate
Mamat, C.; Flemming, A.; Köckerling, M.
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Crystals 2(2012), 90-95
DOI: 10.3390/cryst2010090
ISSN: 2073-4352
The Synthesis and Molecular Structure of 2-(4-Methoxybenzyl)-4-nitro-2H-indazole
Ebert, K.; Köckerling, M.; Mamat, C.
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Crystals 2(2012), 176-181
DOI: 10.3390/cryst2020176
Specific targeting of hypoxic tumor tissue with nitroimidazole-peptide conjugates
Splith, K.; Bergmann, R.; Pietzsch, J.; Neundorf, I.
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ChemMedChem 7(2012), 57-61
DOI: 10.1002/cmdc.201100401
Pyrrolovesamicols - Synthesis, structure and VAChT binding of two 4-fluorobenzoyl regioisomers
Wenzel, B.; Li, Y.; Kraus, W.; Sorger, D.; Sabri, O.; et al. (7 authors)
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Bioorganic & Medicinal Chemistry Letters 22(2012), 2163-2166
DOI: 10.1016/j.bmcl.2012.01.127
The Molecular Structure of 1,2:5,6-Di-O-isopropylidene-3-O-toluenesulfonyl-a-D-glucofuranose
Mamat, C.; Peppel, T.; Köckerling, M.
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Crystals 2(2012), 105-109
DOI: 10.3390/cryst2010105
ISSN: 2073-4352
Imaging of the brain serotonin transporters (SERT) with 18F-labelled fluoromethyl-McN5652 and PET in humans
Hesse, S.; Brust, P.; Mäding, P.; Becker, G.-A.; Seese, A.; et al. (17 authors)
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European Journal of Nuclear Medicine and Molecular Imaging 39(2012)6, 1001-1011
DOI: 10.1007/s00259-012-2078-z
Development of radioligands for α7-nAChR imaging with positron emission tomography
Brust, P.; Peters, D.; Deuther-Conrad, W.
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Current Drug Targets 13(2012)5, 594-601
DOI: 10.2174/138945012800398955
ISSN: 1389-4501
Synthesis, radiofluorination and pharmacological evaluation of fluoromethyl substituted spirocyclic PET tracers for labeling of σ1 receptors in the central nervous system and comparison with longer homologues
Maisonial, A.; Grosse Maestrup, E.; Wiese, C.; Hiller, A.; Schepmann, D.; et al. (9 authors)
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Bioorganic & Medicinal Chemistry 20(2012), 257-269
DOI: 10.1016/j.bmc.2011.11.002
Radiosynthesis and Radiotracer Properties of a 7-(2-[F-18]Fluoroethoxy)-6-methoxy-pyrrolidinylquinazoline for Imaging of Phosphodiesterase 10A with PET
Funke, U.; Deuther-Conrad, W.; Schwan, G.; Maisonial, A.; Scheunemann, M.; et al. (9 authors)
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Pharmaceuticals 5(2012)2, 169-188
DOI: 10.3390/ph5020169
ISSN: 1424-8247
Site-selective radiolabeling of peptides by 18F-fluorobenzoylation with [18F]SFB in solution and on solid phase - a comparative study
Kuchar, M.; Pretze, M.; Knieß, T.; Steinbach, J.; Pietzsch, J.; et al. (6 authors)
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Amino Acids 43(2012), 1431-1443
DOI: 10.1007/s00726-012-1216-z
Effect of leukotriene inhibitors on evolution of experimental brain contusions
Voigt, C. L. M.; Donat, C. K.; Härtig, W.; Förschler, A.; Arendt, T.; et al. (7 authors)
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Neuropathology and Applied Neurobiology 38(2012)4, 354-366
DOI: 10.1111/j.1365-2990.2011.01211.x
Radiosynthesis of a 18F-labeled 2,3-diarylsubstituted indole via McMurry coupling for functional characterization of cyclooxygenase-2 (COX-2) in vitro and in vivo
Kniess, T.; Laube, M.; Bergmann, R.; Graf, F.; Steinbach, J.; et al. (7 authors)
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Bioorganic & Medicinal Chemistry 20(2012), 3410-3421
DOI: 10.1016/j.bmc.2012.04.022
2011
Suitability of bilateral filtering for edge-preserving noise reduction in PET
Hofheinz, F.; Langner, J.; Beuthien-Baumann, B.; Oehme, L.; Steinbach, J.; et al. (7 authors)
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EJNMMI Research 1(2011)23
DOI: 10.1186/2191-219X-1-23
Synthesis of an 18F-labeled cyclin-dependent kinase-2 inhibitor
Svensson, F.; Kniess, T.; Bergmann, R.; Pietzsch, J.; Wuest, F.
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Journal of Labelled Compounds and Radiopharmaceuticals 54(2011), 769-774
DOI: 10.1002/jlcr.1922
S100A2 in cancerogenesis: a friend or a foe?
Wolf, S.; Haase-Kohn, C.; Pietzsch, J.
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Amino Acids 41(2011), 849-861
DOI: 10.1007/s00726-010-0623-2
S100 proteins in health and disease
Pietzsch, J.
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Amino Acids 41(2011), 755-760
DOI: 10.1007/s00726-010-0816-8
Influence of storage on the position of the germinal disc in the fertilized unincubated chicken egg
Burkhardt, A.; Meister, S.; Bergmann, R.; Koch, E.
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Poultry Science 90(2011), 2169-2173
DOI: 10.3382/ps.2010-01179
ISSN: 0032-5791
Synthesis, colloidal stability and 64Cu labeling of iron oxide nanoparticles bearing different macrocyclic ligands
Barreto, J. A.; Matterna, M.; Graham, B.; Stephan, H.; Spiccia, L.
- New Journal of Chemistry 35(2011), 2705-2712
Copper-mediated cross-linking of S100A4, but not of S100A2, results in proinflammatory effects in melanoma cells
Haase-Kohn, C.; Wolf, S.; Lenk, J.; Pietzsch, J.
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Biochemical and Biophysical Research Communications 413(2011), 494-498
DOI: 10.1016/j.bbrc.2011.08.132
Phosphopeptides with improved cellular uptake properties as ligands for the polo-box domain of polo-like kinase 1
Richter, S.; Neundorf, I.; Loebner, K.; Gräber, M.; Berg, T.; et al. (9 authors)
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Bioorganic & Medicinal Chemistry Letters 21(2011), 4686-4689
DOI: 10.1016/j.bmcl.2011.06.103
Comparison of dopamine turnover, dopamine influx constant and activity ratio of striatum and occipital brain with F-18-dopa brain PET in normal controls and patients with Parkinson's disease
Oehme, L.; Perick, M.; Beuthien-Baumann, B.; Wolz, M.; Storch, A.; et al. (11 authors)
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European Journal of Nuclear Medicine and Molecular Imaging 38(2011), 1550-1559
DOI: 10.1007/s00259-011-1819-8
ISSN: 1619-7070
Impact of functionalized coligands on the pharmacokinetics of 99mTc(III) ‘4+1’ mixed-ligand complexes conjugated to bombesin
Künstler, J.-U.; Bergmann, R.; Gniazdowska, E.; Kozminski, P.; Walther, M.; et al. (6 authors)
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Journal of Inorganic Biochemistry 105(2011), 1383-1390
DOI: 10.1016/j.jinorgbio.2011.07.002
Neue Entwicklungen in der PET/CT Hybridbildgebung: Nutzen für die Strahlentherapie?
Hofheinz, F.; Perrin, R.; van den Hoff, J.; Zips, D.
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Der Nuklearmediziner 34(2011), 79-87
DOI: 10.1055/s-0031-1280770
Radiolabeling of phosphatidylserine-binding peptides with prosthetic groups N-[6-(4-[18F]fluorobenzylidene)aminooxyhexyl]maleimide ([18F]FBAM) and N-succinimidyl-4-[18F]fluorobenzoate ([18F]SFB)
Kapty, J.; Kniess, T.; Wuest, F.; Mercer, J. R.
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Applied Radiation and Isotopes 69(2011), 1218-1225
DOI: 10.1016/j.apradiso.2011.05.012
ISSN: 0969-8043
Leitlinie für PET und SPECT–Untersuchungen von Hirntumoren mit radioaktiv markierten Aminosäuren
Langen, K.-J.; Bartenstein, P.; Brust, P.; Coenen, H. H.; Drzezga, A.; et al. (12 authors)
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Nuklearmedizin 50(2011)4, 167-173
DOI: 10.3413/nuk-2011041
Maleimido-Functionalized NOTA Derivatives as Bifunctional Chelators for Site-Specific Radiolabeling
Förster, C.; Schubert, M.; Pietzsch, H.-J.; Steinbach, J.
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Molecules 16(2011), 5228-5240
DOI: 10.3390/molecules16065228
ISSN: 1420-3049
Long-Acting Lipidated Analogue of Human Pancreatic Polypeptide Is Slowly Released into Circulation
Bellmann-Sickert, K.; Elling, C. E.; Madsen, A. N.; Little, P. B.; Lundgren, K.; et al. (10 authors)
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Journal of Medicinal Chemistry 54(2011)8, 2658-2667
DOI: 10.1021/jm101357e
ISSN: 0022-2623
Synthesis, characterization and biological evaluation of [188Re(N)(cys∼)(PNP)]+/0 mixed-ligand complexes as prototypes for the development of 188Re(N)-based target-specific radiopharmaceuticals
Thieme, S.; Agostini, S.; Bergmann, R.; Pietzsch, J.; Pietzsch, H.-J.; et al. (9 authors)
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Nuclear Medicine and Biology 38(2011), 399-415
DOI: 10.1016/j.nucmedbio.2010.09.006
Feasibility and performance of novel software to quantify metabolically active volumes and 3D partial volume corrected SUV and metabolic volumetric products of spinal bone marrow metastases on 18F-FDG-PET/CT.
Torigian, D. A.; Lopez, R. F.; Alapati, S.; Bodapati, G.; Hofheinz, F.; et al. (8 authors)
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Hellenic Journal of Nuclear Medicine 14(2011)1, 8-14
ISSN: 1108-1430
Visualization of the focus in congenital hyperinsulinism by intraoperative sonography
von Rohden, L.; Mohnike, K.; Mau, H.; Eberhard, T.; Mohnike, W.; et al. (10 authors)
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Seminars in Pediatric Surgery 20(2011)1, 28-31
DOI: 10.1053/j.sempedsurg.2010.10.011
ISSN: 1055-8586
Cathepsin S inhibitors: WO2010070615
Löser, R.
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Expert Opinion on Therapeutic Patents 21(2011)4, 585-591
DOI: 10.1517/13543776.2011.550574
ISSN: 1354-3776
Synthesis and evaluation of 1,5-diaryl-substituted tetrazoles as novel selective cyclooxygenase-2 (COX-2) inhibitors
Al-Hourani, B. J.; Sharma, S. K.; Mane, J. Y.; Tuszynski, J.; Baracos, V.; et al. (9 authors)
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Bioorganic & Medicinal Chemistry Letters 21(2011), 1823-1826
DOI: 10.1016/j.bmcl.2011.01.057
ISSN: 0960-894X
Imidazole Containing Bispidine Ligands: Synthesis, Structure and Cu(II)-Complexation
Walther, M.; Matterna, M.; Juran, S.; Fähnemann, S.; Stephan, H.; et al. (7 authors)
- Zeitschrift für Naturforschung Section B - A Journal of Chemical Sciences 66b(2011), 721-728
Expression, purification and fluorine-18 radiolabeling of recombinant S100A4: a potential probe for molecular imaging of receptor for advanced glycation endproducts in vivo?
Wolf, S.; Haase-Kohn, C.; Lenk, J.; Hoppmann, S.; Bergmann, R.; et al. (7 authors)
- Amino Acids 41(2011), 809-820
Zwei oder vier Stunden [18F]FMISO-PET in Kopf-Hals-Karzinomen: Wann ist der Bildkontrast am höchsten?
Abolmaali, N.; Haase, R.; Koch, A.; Zips, D.; Steinbach, J.; et al. (8 authors)
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Nuklearmedizin 50(2011), 22-27
DOI: 10.3413/nukmed-00328-10-07
Intraoperative Sonography: A Technique for Localizing Focal Forms of Congenital Hyperinsulinism in the Pancreas
von Rohden, L.; Mohnike, K.; Mau, H.; Eberhard, T.; Mohnike, W.; et al. (10 authors)
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Ultraschall in der Medizin 32(2011), 74-80
DOI: 10.1055/s-0029-1245598
A 18F-labeled Fluorobutyl-substituted spirocyclic piperidine derivative as a selective radioligand for PET imaging of sigma1 receptors
Maisonial, A.; Große Maestrup, E.; Fischer, S.; Hiller, A.; Scheunemann, M.; et al. (11 authors)
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ChemMedChem 6(2011), 1401-1410
DOI: 10.1002/cmdc.201100108
A Novel Tetrabranched Neurotensin(8-13) Cyclam Derivative: Synthesis, 64Cu-Labeling and Biological Evaluation
Röhrich, A.; Bergmann, R.; Kretzschmann, A.; Noll, S.; Steinbach, J.; et al. (7 authors)
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Journal of Inorganic Biochemistry 105(2011), 821-832
DOI: 10.1016/j.jinorgbio.2011.02.011
Nanomaterials: applications in cancer imaging and therapy
Barreto, J. A.; O'Malley, W.; Kubeil, M.; Graham, B.; Stephan, H.; et al. (6 authors)
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Advanced Materials 23(2011)12, H18-H40
DOI: 10.1002/adma.201190041
Synthesis, structure determination and (radio-) fluorination of novel functionalized phosphanes suitable for the traceless Staudinger ligation
Mamat, C.; Franke, M.; Peppel, T.; Köckerling, M.; Steinbach, J.
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Tetrahedron 67(2011), 4521-4529
DOI: 10.1016/j.tet.2011.04.091
Synthesis and biological evaluation of new [Tc(N)(PS)]-based mixed-ligand compounds useful in design of target-specific radiopharmaceuticas: the 2-methoxyphenylpiperazine dithiocarbamate derivatives as example
Bolzati, C.; Salvarese, N.; Carta, D.; Refosco, F.; Dolmella, A.; et al. (8 authors)
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Journal of Biological Inorganic Chemistry 16(2011), 137-155
DOI: 10.1007/s00775-010-0712-4
[18F]1-(3-fluoropropyl)piperazines as model compounds for the radiofluorination of pyrido[2,3-d]pyrimidines
Grosse-Gehling, P.; Wuest, F. R.; Peppel, T.; Köckerling, M.; Mamat, C.
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Radiochimica Acta 99(2011), 365-373
DOI: 10.1524/ract.2011.1834
Synthesis and biological evaluation of novel 4-benzylpiperazine ligands for sigma-1 receptor imaging
Li, Z.-J.; Ren, H.-Y.; Cui, M.-C.; Deuther-Conrad, W.; Tang, R.-K.; et al. (9 authors)
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Bioorganic & Medicinal Chemistry 19(2011)9, 2911-2917
DOI: 10.1016/j.bmc.2011.03.037
Cross-Coupling Reactions as Valuable Tool for the Preparation of PET Radiotracers
Pretze, M.; Große-Gehling, P.; Mamat, C.
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Molecules 16(2011), 1129-1165
DOI: 10.3390/molecules16021129
In vitro binding profile and radiosynthesis of a novel 18F-labeled azaspirovesamicol analog as potential ligand for imaging of the vesicular acetylcholine transporter
Wenzel, B.; Hiller, A.; Fischer, S.; Sorger, D.; Deuther-Conrad, W.; et al. (9 authors)
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Journal of Labelled Compounds and Radiopharmaceuticals 54(2011), 426-432
DOI: 10.1002/jlcr.1891
High regiocontrol in the nucleophilic ring opening of 1-aralkyl-3,4-epoxypiperidines with amines – A short-step synthesis of 4-fluorobenzyltrozamicol and novel anilidopiperidines
Scheunemann, M.; Hennig, L.; Funke, U.; Steinbach, J.
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Tetrahedron 67(2011), 3448-3456
DOI: 10.1016/j.tet.2011.03.045
Assessment of alpha 7 nicotinic acetylcholine receptor availability in juvenile pig brain with [18F]NS10743
Deuther-Conrad, W.; Fischer, S.; Hiller, A.; Becker, G.; Cumming, P.; et al. (10 authors)
- European Journal of Nuclear Medicine and Molecular Imaging 38(2011)8, 1541-1549
Automated radiosynthesis of the thiol-reactive labeling agent N-[6-(4-[18F]fluorobenzylidene)aminooxyhexyl]maleimide ([18F]FBAM)
Knieß, T.; Kuchar, M.; Pietzsch, J.
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Applied Radiation and Isotopes 69(2011), 1226-1230
DOI: 10.1016/j.apradiso.2011.03.043
Synthesis, pharmacological activity and structure affinity relationships of spirocyclic σ1 receptor ligands with a (2-fluoroethyl) residue in 3-position
Große Maestrup, E.; Wiese, C.; Schepmann, D.; Brust, P.; Wünsch, B.
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Bioorganic & Medicinal Chemistry 19(2011), 393-405
DOI: 10.1016/j.bmc.2010.11.013
The serotonin transporter availability in untreated early-onset and late-onset patients with obsessive-compulsive disorder
Hesse, S.; Stengler, K.; Regenthal, R.; Patt, M.; Becker, G.-A.; et al. (15 authors)
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International Journal of Neuropsychopharmacology 14(2011), 1-12
DOI: 10.1017/S1461145710001604
Molecular imaging of σ receptors: synthesis and evaluation of the potent σ1 selective radioligand [18F]fluspidine
Fischer, S.; Wiese, C.; Grosse Maestrup, E.; Hiller, A.; Deuther-Conrad, W.; et al. (10 authors)
- European Journal of Nuclear Medicine and Molecular Imaging 38(2011)3, 540-551
Traumatic Brain Injury Elicits Similar Alterations in α7 Nicotinic Receptor Density in Two Different Experimental Models
Hoffmeister, P.-G.; Donat, C. K.; Schuhmann, M. U.; Voigt, C.; Walter, B.; et al. (9 authors)
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Neuromolecular Medicine 13(2011)1, 44-53
DOI: 10.1007/s12017-010-8136-4
ISSN: 1535-1084
Enantioselective σ1 receptor binding and biotransformation of the spirocyclic PET tracer 1’-Benzyl-3-(3-fluoropropyl)-3H-spiro[[2]benzofuran-1,4’-piperidine]
Wiese, C.; Große Maestrup, E.; Schepmann, D.; Grimme, S.; Humpf, H.-U.; et al. (7 authors)
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Chirality 23(2011), 148-154
DOI: 10.1002/chir.20893
Design, Synthesis and Preliminary in vitro and in vivo Pharmacological Evaluation of 2-{4-[4-(2,5-disubstituted thiazolyl)phenylethyl] piperazin-1-yl}-1,8-naphthyridine-3- carbonitriles as Atypical Antipsychotic Agents
Chandra Sekhar, K. V. G.; Rao, V. S.; Deuther-Conrad, W.; Reddy, A. S.; Brust, P.; et al. (6 authors)
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Journal of Enzyme Inhibition And Medicinal Chemistry 26(2011)4, 561-568
DOI: 10.3109/14756366.2010.537658
Implementation of 89Zr production and in vivo imaging of B-cells in mice with 89Zr-labeled anti B-cell antibodies by small animal PET/CT
Walther, M.; Gebhardt, P.; Grosse-Gehling, P.; Würbach, L.; Irmler, I.; et al. (11 authors)
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Applied Radiation and Isotopes 69(2011), 852-857
DOI: 10.1016/j.apradiso.2011.02.040
2010
Positron emission tomography 2008 in Germany: Results of the query and current status
Kotzerke, J.; Oehme, L.; Lindner, O.; Hellwig, D.; Bartenstein, P.; et al. (19 authors)
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Nuklearmedizin 49(2010)2, 58-64
DOI: 10.3413/nukmed-0203
ISSN: 0029-5566
Combined correction of recovery effect and motion blur for SUV quantification of solitary pulmonary nodules in FDG PET/CT
Apostolova, I.; Wiemker, R.; Paulus, T.; Kabus, S.; Dreilich, T.; et al. (11 authors)
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European Radiology 20(2010)8, 1868-1877
DOI: 10.1007/s00330-010-1747-1
ISSN: 0938-7994
Modulation of Adrenal Aldosterone Release by Oxidative Modification of Low-Density Lipoprotein
Ansurudeen, I.; Pietzsch, J.; Graessler, J.; Ehrhart-Bornstein, M.; Saha, S.; et al. (7 authors)
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American Journal of Hypertension 23(2010)10, 1061-1068
DOI: 10.1038/ajh.2010.118
ISSN: 0895-7061
Identification of transport processes in bioirrigated muddy sediments by [18F]fluoride PET (Positron Emission Tomography)
Roskosch, A.; Lewandowski, J.; Bergmann, R.; Wilke, F.; Brenner, W.; et al. (6 authors)
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Applied Radiation and Isotopes 68(2010)6, 1094-1097
DOI: 10.1016/j.apradiso.2010.02.004
Noncovalent Tripeptidyl Benzyl- and Cyclohexyl-Amine Inhibitors of the Cysteine Protease Caspase-1
Löser, R.; Abbenante, G.; Madala, P. K.; Halili, M.; Le, G. T.; et al. (6 authors)
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Journal of Medicinal Chemistry 53(2010), 2651-2655
DOI: 10.1021/jm901790w
Antimalarial activity of azadipeptide nitriles
Löser, R.; Gut, J.; Rosenthal, P. J.; Frizler, M.; Gütschow, M.; et al. (6 authors)
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Bioorganic & Medicinal Chemistry Letters 20(2010), 252-255
DOI: 10.1016/j.bmcl.2009.10.122
Sugar-decorated dendritic nanocarriers: Encapsulation and release of the octahedral rhenium cluster complex [Re6S8(OH)6]4-
Kubeil, M.; Stephan, H.; Pietzsch, H.-J.; Geipel, G.; Appelhans, D.; et al. (11 authors)
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Chemistry - An Asian Journal 5(2010), 2507-2514
DOI: 10.1002/asia.201000284
Comparison of the stability of Y-90-, Lu-177- and Ga-68- labeled human serum albumin microspheres (DOTA-HSAM)
Wunderlich, G.; Schiller, E.; Bergmann, R.; Pietzsch, H.-J.
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Nuclear Medicine and Biology 37(2010), 861-867
DOI: 10.1016/j.nucmedbio.2010.05.004
The traceless Staudinger ligation with fluorine-18: a novel and versatile labeling technique for the synthesis of PET-radiotracers
Pretze, M.; Wuest, F.; Peppel, T.; Köckerling, M.; Mamat, C.
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Tetrahedron Letters 51(2010), 6410-6414
DOI: 10.1016/j.tetlet.2010.09.134
Preparation, 99mTc-labeling and biodistribution studies of a PNA oligomer containing a new ligand derivative of 2,2′-dipicolylamine
Gasser, G.; Jäger, K.; Zenker, M.; Bergmann, R.; Steinbach, J.; et al. (7 authors)
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Journal of Inorganic Biochemistry 104(2010), 1133-1140
DOI: 10.1016/j.jinorgbio.2010.06.011
Accessible silanol sites - beneficial for the RP-HPLC separation of constitutional and diastereomeric azaspirovesamicol isomers
Wenzel, B.; Fischer, S.; Brust, P.; Steinbach, J.
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Journal of Chromatography A 1217(2010), 7884-7890
DOI: 10.1016/j.chroma.2010.10.061
A novel Dibenzoazacyclooctyne precursor in regioselective Copper-free click chemistry. An innovative 3-step synthesis.
Starke, F.; Walther, M.; Pietzsch, H.-J.
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ARKIVOC (2010), 350-359
ISSN: 1551-7012
Synthesis and Radiofluorination of Iodophenyl Esters as Tool for the Traceless Staudinger Ligation
Pretze, M.; Flemming, A.; Köckerling, M.; Mamat, C.
- Zeitschrift für Naturforschung Section B - A Journal of Chemical Sciences 65(2010), 1128-1136
3D QSAR study, synthesis and in vitro evaluation of (+)-5-FBVM as potential PET radioligand for the Vesicular AcetylCholine Transporter (VAChT)
Kovac, M.; Mavel, S.; Deuther-Conrad, W.; Méheux, N.; Glöckner, J.; et al. (10 authors)
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Bioorganic & Medicinal Chemistry 18(2010), 7659-7667
DOI: 10.1016/j.bmc.2010.08.028
A new hexanuclear rhenium cluster complex with six terminal acetate ligands: Synthesis, structure, and properties of K4[Re6S8(CH3COO)6]·8H2O
Brylev, K. A.; Mironov, Y. V.; Fedorov, V. E.; Kim, S.-J.; Pietzsch, H.-J.; et al. (8 authors)
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Inorganica Chimica Acta 363(2010)11, 2686-2691
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Novel 99mTc '4 + 1' peptide conjugates: Tuning the biodistribution by variation of coligands
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European Journal of Medicinal Chemistry 45(2010), 3645-3655
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Eph Receptors and Ephrin Ligands: Important Players in Angiogenesis and Tumor Angiogenesis
Mosch, B.; Reissenweber, B.; Neuber, C.; Pietzsch, J.
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Journal of Oncology 2010(2010), 135285
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Cyclin-Dependent Kinase 4/6 (Cdk4/6) Inhibitors: Perspectives in Cancer Therapy and Imaging
Graf, F.; Mosch, B.; Koehler, L.; Bergmann, R.; Wuest, F.; et al. (6 authors)
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Mini-Reviews in Medicinal Chemistry 10(2010), 527-539
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Synthesis and biological evaluation of a radioiodinated spiropiperidine ligand as a potential σ1 receptor imaging agent
Chen, R.-Q.; Li, Y.; Zhang, Q.-Y.; Jia, H.-M.; Deuther-Conrad, W.; et al. (10 authors)
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Journal of Labelled Compounds and Radiopharmaceuticals 53(2010), 569-574
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Design, Synthesis and in Vitro Biological Evaluation of Reference Compounds of 123I and 99Tcm Labeled Indole Radiotracers for σ2 Receptor Imaging
Li, Y.; Jia, H.-M.; Deuther-Conrad, W.; Brust, P.; Steinbach, J.; et al. (6 authors)
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Synthesis of neurotensin(8-13)-phosphopeptide heterodimers via click chemistry
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Bioorganic & Medicinal Chemistry Letters 20(2010), 3306-3309
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Effects of lateral fluid percussion injury on cholinergic markers in the newborn piglet brain
Donat, C. K.; Walter, B.; Kayser, T.; Deuther-Conrad, W.; Schliebs, R.; et al. (9 authors)
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International Journal of Developmental Neuroscience 28(2010), 31-38
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Alterations of cholinergic receptors and the vesicular acetylcholine transporter after lateral fluid percussion injury in newborn piglets
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Neuropathology and Applied Neurobiology 36(2010), 225-236
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Novel Indole Derivatives as Potential Imaging Agents for Alzheimers Disease
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Bulletin of the Korean Chemical Society 31(2010)1, 177-180
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Crystal structure of N-benzyl-4-fluorobenzamide, C14H12FNO, at 173 K
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Zeitschrift für Kristallographie - New Crystal Structures 225(2010), 345-346
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Iodine-124: A Promising Positron Emitter for Organic PET Chemistry
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Molecules 15(2010), 2686-2718
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Efficient preparation of 99mTc(III) 4+1 mixed-ligand complexes for peptide labeling with high specific activity
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Applied Radiation and Isotopes 68(2010), 1728-1733
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Enantioseparation of vesamicol and novel vesamicol analogs by high-performance liquid chromatography on different chiral stationary phases
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Journal of Chromatography A 1217(2010), 3855-3862
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Radiosynthesis and radiopharmacological evaluation of cyclin-dependent kinase 4 (Cdk4) inhibitors
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European Journal of Medicinal Chemistry 45(2010), 727-737
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Scavenger receptors are associated with cellular interactions of S100A12 in vitro and in vivo
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International Journal of Biochemistry & Cell Biology 42(2010), 651-661
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Effects of posture on regional pulmonary blood flow in rats as measured by PET
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Journal of Applied Physiology 108(2010), 422-429
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Comment on "Developing DCE-CT to Quantify Intra-Tumor Heterogeneity in Breast Tumors With Differing Angiogenic Phenotype"
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IEEE Transactions on Medical Imaging 29(2010)4, 1088-1092
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Effects of cold sphere walls in PET phantom measurements on the volume reproducing threshold
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Physics in Medicine and Biology 55(2010), 1099-1113
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Improved Multimodality Imaging Using Alginate Molding in Xenograft Tumor Models
Strobel, K.; Bergmann, R.; Meister, S.; van den Hoff, J.; Pietzsch, J.
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Journal of Magnetic Resonance Imaging 31(2010), 747-752
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2009
Recent Application of Click Chemistry for the Synthesis of Radiotracers for Molecular Imaging
Mamat, C.; Ramenda, T.; Wuest, F.
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