Publications of Institute of Radiopharmaceutical Cancer Research - Year 2019
10 Publications2019
Radiosynthesis and Biological Investigation of a Novel Fluorine-18 Labeled Benzoimidazotriazine- based Radioligand for Imaging of Phosphodiesterase 2A with Positron Emission Tomography
Ritawidya, R.; Wenzel, B.; Teodoro, R.; Toussaint, M.; Kranz, M.; et al. (10 authors)
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Molecules 24(2019)22, 4149
DOI: 10.3390/molecules24224149
One-step radiosynthesis of the MCTs imaging agent [18F]FACH by aliphatic 18F-labelling of a methylsulfonate precursor containing an unprotected carboxylic acid group
Sadeghzadeh, M.; Moldovan, R.-P.; Teodoro, R.; Brust, P.; Wenzel, B.
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Scientific Reports 9(2019), 18890
DOI: 10.1038/s41598-019-55354-w
Structure–Affinity Relationships of Fluorinated Spirocyclic Sigma2 Receptor Ligands with an Exocyclic Benzylamino Moiety
Bergkemper, M.; Kronenberg, E.; Schepmann, D.; Ludwig, F.-A.; Brust, P.; et al. (6 authors)
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ChemMedChem 14(2019), 1392-1402
DOI: 10.1002/cmdc.201900284
¹⁸F-Labeled benzylpiperazine derivatives as highly selective ligands for imaging σ1 receptor with positron emission tomography
Ye, J.; Wang, L.; Deuther-Conrad, W.; Chen, Y.; Zhang, X.; et al. (9 authors)
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Journal of Labelled Compounds and Radiopharmaceuticals 62(2019)8, 425-437
DOI: 10.1002/jlcr.3738
Synthesis and in vitro evaluation of 8-pyridinyl substituted benzo[e]imidazo[2,1-c][1,2,4]triazines as phosphodiesterase 2A (PDE2A) inhibitors
Ritawidya, R.; Ludwig, F.-A.; Briel, D.; Brust, P.; Scheunemann, M.
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Molecules 24(2019)15, 2791
DOI: 10.3390/molecules24152791
SPECT-Untersuchungen mit dem 123 I-markierten Dopamintransporter-Liganden FP-CIT (DaTSCAN):DGN-Handlungsempfehlung (S1-Leitlinie)
Tatsch, K.; Buchert, R.; Bartenstein, P.; Barthel, H.; Boecker, H.; et al. (17 authors)
- Nuklearmedizin 58(2019)1, 5-16
In vitro and in vivo Human Metabolism of (S)-[18F]Fluspidine – a Radioligand for Imaging σ1 Receptors with Positron Emission Tomography (PET)
Ludwig, F.-A.; Fischer, S.; Houska, R.; Hoepping, A.; Deuther-Conrad, W.; et al. (15 authors)
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Frontiers in Pharmacology 10(2019), 534
DOI: 10.3389/fphar.2019.00534
Development and radiosynthesis of the first 18F-labeled inhibitor of monocarboxylate transporters (MCTs)
Sadeghzadeh, M.; Moldovan, R.-P.; Fischer, S.; Wenzel, B.; Ludwig, F.-A.; et al. (14 authors)
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Journal of Labelled Compounds and Radiopharmaceuticals 62(2019)8, 411-424
DOI: 10.1002/jlcr.3739
Targeting cyclic nucleotide phosphodiesterase 5 (PDE5) in brain: Toward the development of a PET radioligand labeled with fluorine-18
Wenzel, B.; Liu, J.; Dukic-Stefanovic, S.; Deuther-Conrad, W.; Teodoro, R.; et al. (10 authors)
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Bioorganic Chemistry 86(2019), 346-362
DOI: 10.1016/j.bioorg.2019.01.037
Studies towards the development of a PET radiotracer for imaging of the P2Y1 receptors in the brain: synthesis, 18F-labeling and preliminary biological evaluation
Moldovan, R.-P.; Wenzel, B.; Teodoro, R.; Neumann, W.; Dukic-Stefanovic, S.; et al. (9 authors)
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European Journal of Medicinal Chemistry (2019), 142-159
DOI: 10.1016/j.ejmech.2019.01.006
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