Publications of Institute of Radiopharmaceutical Cancer Research - Year 2017
17 Publications2017
Maternal immune activation results in complex microglial transcriptome signature in the adult offspring that is reversed by minocycline treatment
Mattei, D.; Ivanov, A.; Ferrai, C.; Jordan, P.; Guneykaya, D.; et al. (21 authors)
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Translational Psychiatry 7(2017)e1120, 1-13
DOI: 10.1038/tp.2017.80
PET Imaging Evaluation of Four sigma1 Radiotracers in Nonhuman Primates
Baum, E.; Cai, Z.; Bois, F.; Holden, D.; Lin, S.-F.; et al. (16 authors)
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Journal of Nuclear Medicine 58(2017)6, 982
DOI: 10.2967/jnumed.116.188052
1‑(4‑[18F]Fluorobenzyl)-4-[(tetrahydrofuran-2-yl)methyl]piperazine: A Novel Suitable Radioligand with Low Lipophilicity for Imaging σ1 Receptors in the Brain
He, Y.; Xie, F.; Ye, J.; Deuther-Conrad, W.; Cui, B.; et al. (12 authors)
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Journal of Medicinal Chemistry 60(2017), 4161-4172
DOI: 10.1021/acs.jmedchem.6b01723
18F-Labeled indole-based analogs as highly selective radioligands for imaging sigma-2 receptors in the brain
Wang, L.; Ye, J.; He, Y.; Deuther-Conrad, W.; Zhang, J.; et al. (11 authors)
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Bioorganic & Medicinal Chemistry 25(2017), 3792-3802
DOI: 10.1016/j.bmc.2017.05.019
Synthesis and in vitro evaluation of 5-substituted benzovesamicol analogs containing N-substituted amides as potential positron emission tomography tracers for the vesicular acetylcholine transporter
Roslin, S.; de Rosa, M.; Deuther-Conrad, W.; Eriksson, J.; Odell, L. R.; et al. (8 authors)
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Bioorganic & Medicinal Chemistry 25(2017)19, 5095-5106
DOI: 10.1016/j.bmc.2017.01.041
Radiosynthesis of (S)-[18F]T1: The first PET radioligand for molecular imaging of α3β4 nicotinic acetylcholine receptors
Sarasamkan, J.; Fischer, S.; Deuther-Conrad, W.; Ludwig, F.-A.; Scheunemann, M.; et al. (8 authors)
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Applied Radiation and Isotopes 124(2017), 106-113
DOI: 10.1016/j.apradiso.2017.03.015
Do spiroindolines have the potential to replace vesamicol as lead compound for the development of radioligands targeting the vesicular acetylcholine transporter?
Lindemann, M.; Deuther-Conrad, W.; Moldovan, R.; Sekhar, K. V. G. C.; Brust, P.; et al. (6 authors)
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Bioorganic & Medicinal Chemistry 25(2017)19, 5107-5113
DOI: 10.1016/j.bmc.2017.03.028
Development of highly affine and selective fluorinated cannabinoid receptor type 2 ligands
Moldovan, R.-P.; Hausmann, K.; Deuther-Conrad, W.; Brust, P.
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ACS Medicinal Chemistry Letters (2017), 566-571
DOI: 10.1021/acsmedchemlett.7b00129
Development of Fluorinated Non-Peptidic Ghrelin Receptor Ligands for Potential Use in Molecular Imaging
Moldovan, R.-P.; Els-Heindl, S.; Worm, D. J.; Kniess, T.; Kluge, M.; et al. (9 authors)
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International Journal of Molecular Sciences 18(2017)4, 768
DOI: 10.3390/ijms18040768
PET Imaging of α7 Nicotinic Acetylcholine Receptors: A comparative study of [18F]ASEM and [18F]DBT-10 in non-human primates, and further evaluation of [18F]ASEM in humans
Hillmer, A. T.; Li, S.; Zheng, M.-Q.; Scheunemann, M.; Lin, S.-F.; et al. (17 authors)
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European Journal of Nuclear Medicine and Molecular Imaging 44(2017)6, 1042-1050
DOI: 10.1007/s00259-017-3621-8
Suppressed Fat Appetite after Roux-en-Y Gastric Bypass Surgery Associates with Reduced Brain µ-opioid Receptor Availability in Diet-Induced Obese Male Rats
Hankir, M.; Patt, M.; Patt, J.; Becker, G.; Rullmann, M.; et al. (14 authors)
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Frontiers in Neuroscience 10(2017), 620
Online First (2016) DOI: 10.3389/fnins.2016.00620
Synthesis and in vitro evaluation of new fluorinated quinoline derivatives with high affinity for PDE5: Towards the development of new PET neuroimaging probes
Liu, J.; Maisonial-Besset, A.; Wenzel, B.; Canitrot, D.; Baufond, A.; et al. (8 authors)
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European Journal of Medicinal Chemistry 136(2017), 548-560
DOI: 10.1016/j.ejmech.2017.03.091
Gender Differences in Neural Networks for Color Processing in Mice: A PET/MR Study
Njemanze, P. C.; Kranz, M.; Amend, M.; Wehrl, H.; Brust, P.
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PLOS ONE 12(2017)7, e0179919.
DOI: 10.1371/journal.pone.0179919
Dissociation between brown adipose tissue 18F-FDG uptake and thermogenesis in uncoupling protein deficient mice
Hankir, M. K.; Kranz, M.; Keipert, S.; Andreasen, S.; Kern, M.; et al. (11 authors)
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Journal of Nuclear Medicine 58(2017)7, 1100-1103
DOI: 10.2967/jnumed.116.186460
Synthesis and Preliminary Biological Evaluation of Indol-3-yl-oxoacetamides as Potent Cannabinoid Receptor Type 2 Ligands
Moldovan, R.-P.; Deuther-Conrad, W.; Horti, A. G.; Brust, P.
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Molecules 22(2017)1, 77
DOI: 10.3390/molecules22010077
Gastric Bypass Surgery Recruits a Gut – Striatal Dopamine Pathway to Reduce Fat Appetite in Obese Rats
Hankir, M. K.; Seyfried, F.; Hintschich, C. A.; Diep, T. A.; Kleberg, K.; et al. (17 authors)
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Cell Metabolism 25(2017)2, 335-344
Online First (2016) DOI: 10.1016/j.cmet.2016.12.006
Radiosynthesis and biological evaluation of the new PDE10A radioligand [18F]AQ28A
Wagner, S.; Teodoro, R.; Deuther-Conrad, W.; Kranz, M.; Scheunemann, M.; et al. (11 authors)
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Journal of Labelled Compounds and Radiopharmaceuticals 60(2017)1, 36-48
Online First (2016) DOI: 10.1002/jlcr.3471