Publications of Institute of Radiopharmaceutical Cancer Research - Year 2013
13 Publications2013
Development of fluorinated CB2 receptor agonists for PET studies
Lueg, C.; Schepmann, D.; Günther, R.; Brust, P.; Wünsch, B.
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Bioorganic & Medicinal Chemistry 21(2013), 7481-7498
DOI: 10.1016/j.bmc.2013.09.040
Synthesis, Characterization, and Metabolism Studies of Fluspidine Enantiomers
Holl, K.; Falck, E.; Köhler, J.; Schepmann, D.; Humpf, H.-U.; et al. (7 authors)
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ChemMedChem 8(2013)12, 2047-2056
DOI: 10.1002/cmdc.201300322
Radiofluorination and biological evaluation of N-aryl-oxadiazolyl-propionamides as potential radioligands for PET imaging of cannabinoid CB2 receptors
Teodoro, R.; Moldovan, R.-P.; Lueg, C.; Günther, R.; Donat, C. K.; et al. (10 authors)
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Organic and Medicinal Chemistry Letters 3(2013)11
DOI: 10.1186/2191-2858-3-11
Fully automated radiosynthesis of both enantiomers of [18F]Flubatine under GMP conditions for human application
Patt, M.; Schildan, A.; Habermann, B.; Fischer, S.; Hiller, A.; et al. (13 authors)
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Applied Radiation and Isotopes 80(2013), 7-11
DOI: 10.1016/j.apradiso.2013.05.009
ISSN: 0969-8043
Use of 3-[18F]fluoropropanesulfonyl chloride as prosthetic agent for the radiolabelling of amines: Investigation of precursor molecules, labelling conditions and enzymatic stability of the corresponding sulfonamides
Löser, R.; Fischer, S.; Hiller, A.; Köckerling, M.; Funke, U.; et al. (8 authors)
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Beilstein Journal of Organic Chemistry 9(2013), 1002-1011
DOI: 10.3762/bjoc.9.115
Synthesis and Evaluation of Novel 18F-Labeled Spirocyclic Piperidine Derivatives as σ1 Receptor Ligands for Positron Emission Tomography Imaging
Li, Y.; Wang, X.; Zhang, J.; Deuther-Conrad, W.; Xie, F.; et al. (13 authors)
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Journal of Medicinal Chemistry 56(2013), 3478-3491
DOI: 10.1021/jm301734g
ISSN: 0022-2623
A fluoro versus a nitro derivative - a high-performance liquid chromatography study of two basic analytes with different RP and silica phases as basis for the separation of a positron emission tomography radiotracer
Wenzel, B.; Günther, R.; Brust, P.; Steinbach, J.
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Journal of Chromatography A 1311(2013), 98-105
DOI: 10.1016/j.chroma.2013.08.068
Resistance of brain glucose metabolism to thiopental-induced CNS depression in newborn piglets
Bernd, W.; Eiselt, M.; Cumming, P.; Xiong, G.; Hinz, R.; et al. (8 authors)
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International Journal of Developmental Neuroscience 31(2013), 157-164
DOI: 10.1016/j.ijdevneu.2012.12.008
ISSN: 0736-5748
Radiosynthesis and first evaluation in mice of [18F]NS14490 for molecular imaging of α7 nicotinic acetylcholine receptors
Rötering, S.; Scheunemann, M.; Fischer, S.; Hiller, A.; Peters, D.; et al. (7 authors)
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Bioorganic & Medicinal Chemistry 21(2013), 2635-2642
DOI: 10.1016/j.bmc.2013.02.018
Synthesis and biological evaluation of 18F labeled fluoro-oligo-ethoxylated 4-benzylpiperazine derivatives for sigma-1 receptor imaging
Wang, X.; Li, Y.; Deuther-Conrad, W.; Xie, F.; Chen, X.; et al. (12 authors)
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Bioorganic & Medicinal Chemistry 21(2013)1, 215-222
Online First (2012) DOI: 10.1016/j.bmc.2012.10.038
Leitlinie für die Hirnperfusions-SPECT mit Tc-99m Radiopharmaka / Hirnperfusions-SPECT with 99mTc-labelled Radiopharmaceuticals DGN-Guidance (S1 Guideline)
Kranert, T.; Menzel, C.; Bartenstein, P.; Brust, P.; Coenen, H. H.; et al. (11 authors)
- Nuklearmedizin 5(2013)52, 157-162
Radiosynthesis of racemic and enantiomerically pure (–)-[18F]flubatine – A promising PET radiotracer for neuroimaging of α4β2 nicotinic acetylcholine receptors
Fischer, S.; Hiller, A.; Smits, R.; Hoepping, A.; Funke, U.; et al. (10 authors)
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Applied Radiation and Isotopes 74(2013), 128-136
DOI: 10.1016/j.apradiso.2013.01.002
ISSN: 0969-8043
Design, synthesis, and preliminary in vitro and in vivo pharmacological evaluation of 4-{4-[2-(4-(2-substitutedquinoxalin-3-yl)piperazin-1-yl)ethyl]phenyl}thiazoles as atypical antipsychotic agents
Chandra Sekhar, K. V. G.; Rao, V. S.; Deuther-Conrad, W.; Sridhar, D.; Nagesh, H. N.; et al. (8 authors)
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Medicinal Chemistry Research 22(2013)4, 1660-1673
Online First (2012) DOI: 10.1007/s00044-012-0164-1
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