Publications of Institute of Radiopharmaceutical Cancer Research - Year 2011

43 Publications

2011

Suitability of bilateral filtering for edge-preserving noise reduction in PET

Hofheinz, F.; Langner, J.; Beuthien-Baumann, B.; Oehme, L.; Steinbach, J.; et al. (7 authors)

Synthesis of an 18F-labeled cyclin-dependent kinase-2 inhibitor

Svensson, F.; Kniess, T.; Bergmann, R.; Pietzsch, J.; Wuest, F.

  • Journal of Labelled Compounds and Radiopharmaceuticals 54(2011), 769-774
    DOI: 10.1002/jlcr.1922

S100A2 in cancerogenesis: a friend or a foe?

Wolf, S.; Haase-Kohn, C.; Pietzsch, J.

S100 proteins in health and disease

Pietzsch, J.

Influence of storage on the position of the germinal disc in the fertilized unincubated chicken egg

Burkhardt, A.; Meister, S.; Bergmann, R.; Koch, E.

Synthesis, colloidal stability and 64Cu labeling of iron oxide nanoparticles bearing different macrocyclic ligands

Barreto, J. A.; Matterna, M.; Graham, B.; Stephan, H.; Spiccia, L.

  • New Journal of Chemistry 35(2011), 2705-2712

Copper-mediated cross-linking of S100A4, but not of S100A2, results in proinflammatory effects in melanoma cells

Haase-Kohn, C.; Wolf, S.; Lenk, J.; Pietzsch, J.

Phosphopeptides with improved cellular uptake properties as ligands for the polo-box domain of polo-like kinase 1

Richter, S.; Neundorf, I.; Loebner, K.; Gräber, M.; Berg, T.; et al. (9 authors)

Comparison of dopamine turnover, dopamine influx constant and activity ratio of striatum and occipital brain with F-18-dopa brain PET in normal controls and patients with Parkinson's disease

Oehme, L.; Perick, M.; Beuthien-Baumann, B.; Wolz, M.; Storch, A.; et al. (11 authors)

  • European Journal of Nuclear Medicine and Molecular Imaging 38(2011), 1550-1559
    DOI: 10.1007/s00259-011-1819-8
    ISSN: 1619-7070

Impact of functionalized coligands on the pharmacokinetics of 99mTc(III) ‘4+1’ mixed-ligand complexes conjugated to bombesin

Künstler, J.-U.; Bergmann, R.; Gniazdowska, E.; Kozminski, P.; Walther, M.; et al. (6 authors)

Neue Entwicklungen in der PET/CT Hybridbildgebung: Nutzen für die Strahlentherapie?

Hofheinz, F.; Perrin, R.; van den Hoff, J.; Zips, D.

Radiolabeling of phosphatidylserine-binding peptides with prosthetic groups N-[6-(4-[18F]fluorobenzylidene)aminooxyhexyl]maleimide ([18F]FBAM) and N-succinimidyl-4-[18F]fluorobenzoate ([18F]SFB)

Kapty, J.; Kniess, T.; Wuest, F.; Mercer, J. R.

Leitlinie für PET und SPECT–Untersuchungen von Hirntumoren mit radioaktiv markierten Aminosäuren

Langen, K.-J.; Bartenstein, P.; Brust, P.; Coenen, H. H.; Drzezga, A.; et al. (12 authors)

Maleimido-Functionalized NOTA Derivatives as Bifunctional Chelators for Site-Specific Radiolabeling

Förster, C.; Schubert, M.; Pietzsch, H.-J.; Steinbach, J.

Long-Acting Lipidated Analogue of Human Pancreatic Polypeptide Is Slowly Released into Circulation

Bellmann-Sickert, K.; Elling, C. E.; Madsen, A. N.; Little, P. B.; Lundgren, K.; et al. (10 authors)

  • Journal of Medicinal Chemistry 54(2011)8, 2658-2667
    DOI: 10.1021/jm101357e
    ISSN: 0022-2623

Synthesis, characterization and biological evaluation of [188Re(N)(cys∼)(PNP)]+/0 mixed-ligand complexes as prototypes for the development of 188Re(N)-based target-specific radiopharmaceuticals

Thieme, S.; Agostini, S.; Bergmann, R.; Pietzsch, J.; Pietzsch, H.-J.; et al. (9 authors)

Feasibility and performance of novel software to quantify metabolically active volumes and 3D partial volume corrected SUV and metabolic volumetric products of spinal bone marrow metastases on 18F-FDG-PET/CT.

Torigian, D. A.; Lopez, R. F.; Alapati, S.; Bodapati, G.; Hofheinz, F.; et al. (8 authors)

  • Open Access Logo Hellenic Journal of Nuclear Medicine 14(2011)1, 8-14
    ISSN: 1108-1430

Visualization of the focus in congenital hyperinsulinism by intraoperative sonography

von Rohden, L.; Mohnike, K.; Mau, H.; Eberhard, T.; Mohnike, W.; et al. (10 authors)

Cathepsin S inhibitors: WO2010070615

Löser, R.

Synthesis and evaluation of 1,5-diaryl-substituted tetrazoles as novel selective cyclooxygenase-2 (COX-2) inhibitors

Al-Hourani, B. J.; Sharma, S. K.; Mane, J. Y.; Tuszynski, J.; Baracos, V.; et al. (9 authors)

Imidazole Containing Bispidine Ligands: Synthesis, Structure and Cu(II)-Complexation

Walther, M.; Matterna, M.; Juran, S.; Fähnemann, S.; Stephan, H.; et al. (7 authors)

  • Zeitschrift für Naturforschung Section B - A Journal of Chemical Sciences 66b(2011), 721-728

Expression, purification and fluorine-18 radiolabeling of recombinant S100A4: a potential probe for molecular imaging of receptor for advanced glycation endproducts in vivo?

Wolf, S.; Haase-Kohn, C.; Lenk, J.; Hoppmann, S.; Bergmann, R.; et al. (7 authors)

  • Amino Acids 41(2011), 809-820

Zwei oder vier Stunden [18F]FMISO-PET in Kopf-Hals-Karzinomen: Wann ist der Bildkontrast am höchsten?

Abolmaali, N.; Haase, R.; Koch, A.; Zips, D.; Steinbach, J.; et al. (8 authors)

Intraoperative Sonography: A Technique for Localizing Focal Forms of Congenital Hyperinsulinism in the Pancreas

von Rohden, L.; Mohnike, K.; Mau, H.; Eberhard, T.; Mohnike, W.; et al. (10 authors)

A 18F-labeled Fluorobutyl-substituted spirocyclic piperidine derivative as a selective radioligand for PET imaging of sigma1 receptors

Maisonial, A.; Große Maestrup, E.; Fischer, S.; Hiller, A.; Scheunemann, M.; et al. (11 authors)

A Novel Tetrabranched Neurotensin(8-13) Cyclam Derivative: Synthesis, 64Cu-Labeling and Biological Evaluation

Röhrich, A.; Bergmann, R.; Kretzschmann, A.; Noll, S.; Steinbach, J.; et al. (7 authors)

Nanomaterials: applications in cancer imaging and therapy

Barreto, J. A.; O'Malley, W.; Kubeil, M.; Graham, B.; Stephan, H.; et al. (6 authors)

Synthesis, structure determination and (radio-) fluorination of novel functionalized phosphanes suitable for the traceless Staudinger ligation

Mamat, C.; Franke, M.; Peppel, T.; Köckerling, M.; Steinbach, J.

Synthesis and biological evaluation of new [Tc(N)(PS)]-based mixed-ligand compounds useful in design of target-specific radiopharmaceuticas: the 2-methoxyphenylpiperazine dithiocarbamate derivatives as example

Bolzati, C.; Salvarese, N.; Carta, D.; Refosco, F.; Dolmella, A.; et al. (8 authors)

[18F]1-(3-fluoropropyl)piperazines as model compounds for the radiofluorination of pyrido[2,3-d]pyrimidines

Grosse-Gehling, P.; Wuest, F. R.; Peppel, T.; Köckerling, M.; Mamat, C.

Synthesis and biological evaluation of novel 4-benzylpiperazine ligands for sigma-1 receptor imaging

Li, Z.-J.; Ren, H.-Y.; Cui, M.-C.; Deuther-Conrad, W.; Tang, R.-K.; et al. (9 authors)

Cross-Coupling Reactions as Valuable Tool for the Preparation of PET Radiotracers

Pretze, M.; Große-Gehling, P.; Mamat, C.

In vitro binding profile and radiosynthesis of a novel 18F-labeled azaspirovesamicol analog as potential ligand for imaging of the vesicular acetylcholine transporter

Wenzel, B.; Hiller, A.; Fischer, S.; Sorger, D.; Deuther-Conrad, W.; et al. (9 authors)

  • Journal of Labelled Compounds and Radiopharmaceuticals 54(2011), 426-432
    DOI: 10.1002/jlcr.1891

High regiocontrol in the nucleophilic ring opening of 1-aralkyl-3,4-epoxypiperidines with amines – A short-step synthesis of 4-fluorobenzyltrozamicol and novel anilidopiperidines

Scheunemann, M.; Hennig, L.; Funke, U.; Steinbach, J.

Assessment of alpha 7 nicotinic acetylcholine receptor availability in juvenile pig brain with [18F]NS10743

Deuther-Conrad, W.; Fischer, S.; Hiller, A.; Becker, G.; Cumming, P.; et al. (10 authors)

  • European Journal of Nuclear Medicine and Molecular Imaging 38(2011)8, 1541-1549

Automated radiosynthesis of the thiol-reactive labeling agent N-[6-(4-[18F]fluorobenzylidene)aminooxyhexyl]maleimide ([18F]FBAM)

Knieß, T.; Kuchar, M.; Pietzsch, J.

Synthesis, pharmacological activity and structure affinity relationships of spirocyclic σ1 receptor ligands with a (2-fluoroethyl) residue in 3-position

Große Maestrup, E.; Wiese, C.; Schepmann, D.; Brust, P.; Wünsch, B.

The serotonin transporter availability in untreated early-onset and late-onset patients with obsessive-compulsive disorder

Hesse, S.; Stengler, K.; Regenthal, R.; Patt, M.; Becker, G.-A.; et al. (15 authors)

Molecular imaging of σ receptors: synthesis and evaluation of the potent σ1 selective radioligand [18F]fluspidine

Fischer, S.; Wiese, C.; Grosse Maestrup, E.; Hiller, A.; Deuther-Conrad, W.; et al. (10 authors)

  • European Journal of Nuclear Medicine and Molecular Imaging 38(2011)3, 540-551

Traumatic Brain Injury Elicits Similar Alterations in α7 Nicotinic Receptor Density in Two Different Experimental Models

Hoffmeister, P.-G.; Donat, C. K.; Schuhmann, M. U.; Voigt, C.; Walter, B.; et al. (9 authors)

Enantioselective σ1 receptor binding and biotransformation of the spirocyclic PET tracer 1’-Benzyl-3-(3-fluoropropyl)-3H-spiro[[2]benzofuran-1,4’-piperidine]

Wiese, C.; Große Maestrup, E.; Schepmann, D.; Grimme, S.; Humpf, H.-U.; et al. (7 authors)

Design, Synthesis and Preliminary in vitro and in vivo Pharmacological Evaluation of 2-{4-[4-(2,5-disubstituted thiazolyl)phenylethyl] piperazin-1-yl}-1,8-naphthyridine-3- carbonitriles as Atypical Antipsychotic Agents

Chandra Sekhar, K. V. G.; Rao, V. S.; Deuther-Conrad, W.; Reddy, A. S.; Brust, P.; et al. (6 authors)

Implementation of 89Zr production and in vivo imaging of B-cells in mice with 89Zr-labeled anti B-cell antibodies by small animal PET/CT

Walther, M.; Gebhardt, P.; Grosse-Gehling, P.; Würbach, L.; Irmler, I.; et al. (11 authors)

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