Publications of Institute of Radiopharmaceutical Cancer Research - Year 2011
43 Publications2011
Suitability of bilateral filtering for edge-preserving noise reduction in PET
Hofheinz, F.; Langner, J.; Beuthien-Baumann, B.; Oehme, L.; Steinbach, J.; et al. (7 authors)
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EJNMMI Research 1(2011)23
DOI: 10.1186/2191-219X-1-23
Synthesis of an 18F-labeled cyclin-dependent kinase-2 inhibitor
Svensson, F.; Kniess, T.; Bergmann, R.; Pietzsch, J.; Wuest, F.
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Journal of Labelled Compounds and Radiopharmaceuticals 54(2011), 769-774
DOI: 10.1002/jlcr.1922
S100A2 in cancerogenesis: a friend or a foe?
Wolf, S.; Haase-Kohn, C.; Pietzsch, J.
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Amino Acids 41(2011), 849-861
DOI: 10.1007/s00726-010-0623-2
S100 proteins in health and disease
Pietzsch, J.
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Amino Acids 41(2011), 755-760
DOI: 10.1007/s00726-010-0816-8
Influence of storage on the position of the germinal disc in the fertilized unincubated chicken egg
Burkhardt, A.; Meister, S.; Bergmann, R.; Koch, E.
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Poultry Science 90(2011), 2169-2173
DOI: 10.3382/ps.2010-01179
ISSN: 0032-5791
Synthesis, colloidal stability and 64Cu labeling of iron oxide nanoparticles bearing different macrocyclic ligands
Barreto, J. A.; Matterna, M.; Graham, B.; Stephan, H.; Spiccia, L.
- New Journal of Chemistry 35(2011), 2705-2712
Copper-mediated cross-linking of S100A4, but not of S100A2, results in proinflammatory effects in melanoma cells
Haase-Kohn, C.; Wolf, S.; Lenk, J.; Pietzsch, J.
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Biochemical and Biophysical Research Communications 413(2011), 494-498
DOI: 10.1016/j.bbrc.2011.08.132
Phosphopeptides with improved cellular uptake properties as ligands for the polo-box domain of polo-like kinase 1
Richter, S.; Neundorf, I.; Loebner, K.; Gräber, M.; Berg, T.; et al. (9 authors)
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Bioorganic & Medicinal Chemistry Letters 21(2011), 4686-4689
DOI: 10.1016/j.bmcl.2011.06.103
Comparison of dopamine turnover, dopamine influx constant and activity ratio of striatum and occipital brain with F-18-dopa brain PET in normal controls and patients with Parkinson's disease
Oehme, L.; Perick, M.; Beuthien-Baumann, B.; Wolz, M.; Storch, A.; et al. (11 authors)
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European Journal of Nuclear Medicine and Molecular Imaging 38(2011), 1550-1559
DOI: 10.1007/s00259-011-1819-8
ISSN: 1619-7070
Impact of functionalized coligands on the pharmacokinetics of 99mTc(III) ‘4+1’ mixed-ligand complexes conjugated to bombesin
Künstler, J.-U.; Bergmann, R.; Gniazdowska, E.; Kozminski, P.; Walther, M.; et al. (6 authors)
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Journal of Inorganic Biochemistry 105(2011), 1383-1390
DOI: 10.1016/j.jinorgbio.2011.07.002
Neue Entwicklungen in der PET/CT Hybridbildgebung: Nutzen für die Strahlentherapie?
Hofheinz, F.; Perrin, R.; van den Hoff, J.; Zips, D.
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Der Nuklearmediziner 34(2011), 79-87
DOI: 10.1055/s-0031-1280770
Radiolabeling of phosphatidylserine-binding peptides with prosthetic groups N-[6-(4-[18F]fluorobenzylidene)aminooxyhexyl]maleimide ([18F]FBAM) and N-succinimidyl-4-[18F]fluorobenzoate ([18F]SFB)
Kapty, J.; Kniess, T.; Wuest, F.; Mercer, J. R.
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Applied Radiation and Isotopes 69(2011), 1218-1225
DOI: 10.1016/j.apradiso.2011.05.012
ISSN: 0969-8043
Leitlinie für PET und SPECT–Untersuchungen von Hirntumoren mit radioaktiv markierten Aminosäuren
Langen, K.-J.; Bartenstein, P.; Brust, P.; Coenen, H. H.; Drzezga, A.; et al. (12 authors)
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Nuklearmedizin 50(2011)4, 167-173
DOI: 10.3413/nuk-2011041
Maleimido-Functionalized NOTA Derivatives as Bifunctional Chelators for Site-Specific Radiolabeling
Förster, C.; Schubert, M.; Pietzsch, H.-J.; Steinbach, J.
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Molecules 16(2011), 5228-5240
DOI: 10.3390/molecules16065228
ISSN: 1420-3049
Long-Acting Lipidated Analogue of Human Pancreatic Polypeptide Is Slowly Released into Circulation
Bellmann-Sickert, K.; Elling, C. E.; Madsen, A. N.; Little, P. B.; Lundgren, K.; et al. (10 authors)
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Journal of Medicinal Chemistry 54(2011)8, 2658-2667
DOI: 10.1021/jm101357e
ISSN: 0022-2623
Synthesis, characterization and biological evaluation of [188Re(N)(cys∼)(PNP)]+/0 mixed-ligand complexes as prototypes for the development of 188Re(N)-based target-specific radiopharmaceuticals
Thieme, S.; Agostini, S.; Bergmann, R.; Pietzsch, J.; Pietzsch, H.-J.; et al. (9 authors)
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Nuclear Medicine and Biology 38(2011), 399-415
DOI: 10.1016/j.nucmedbio.2010.09.006
Feasibility and performance of novel software to quantify metabolically active volumes and 3D partial volume corrected SUV and metabolic volumetric products of spinal bone marrow metastases on 18F-FDG-PET/CT.
Torigian, D. A.; Lopez, R. F.; Alapati, S.; Bodapati, G.; Hofheinz, F.; et al. (8 authors)
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Hellenic Journal of Nuclear Medicine 14(2011)1, 8-14
ISSN: 1108-1430
Visualization of the focus in congenital hyperinsulinism by intraoperative sonography
von Rohden, L.; Mohnike, K.; Mau, H.; Eberhard, T.; Mohnike, W.; et al. (10 authors)
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Seminars in Pediatric Surgery 20(2011)1, 28-31
DOI: 10.1053/j.sempedsurg.2010.10.011
ISSN: 1055-8586
Cathepsin S inhibitors: WO2010070615
Löser, R.
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Expert Opinion on Therapeutic Patents 21(2011)4, 585-591
DOI: 10.1517/13543776.2011.550574
ISSN: 1354-3776
Synthesis and evaluation of 1,5-diaryl-substituted tetrazoles as novel selective cyclooxygenase-2 (COX-2) inhibitors
Al-Hourani, B. J.; Sharma, S. K.; Mane, J. Y.; Tuszynski, J.; Baracos, V.; et al. (9 authors)
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Bioorganic & Medicinal Chemistry Letters 21(2011), 1823-1826
DOI: 10.1016/j.bmcl.2011.01.057
ISSN: 0960-894X
Imidazole Containing Bispidine Ligands: Synthesis, Structure and Cu(II)-Complexation
Walther, M.; Matterna, M.; Juran, S.; Fähnemann, S.; Stephan, H.; et al. (7 authors)
- Zeitschrift für Naturforschung Section B - A Journal of Chemical Sciences 66b(2011), 721-728
Expression, purification and fluorine-18 radiolabeling of recombinant S100A4: a potential probe for molecular imaging of receptor for advanced glycation endproducts in vivo?
Wolf, S.; Haase-Kohn, C.; Lenk, J.; Hoppmann, S.; Bergmann, R.; et al. (7 authors)
- Amino Acids 41(2011), 809-820
Zwei oder vier Stunden [18F]FMISO-PET in Kopf-Hals-Karzinomen: Wann ist der Bildkontrast am höchsten?
Abolmaali, N.; Haase, R.; Koch, A.; Zips, D.; Steinbach, J.; et al. (8 authors)
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Nuklearmedizin 50(2011), 22-27
DOI: 10.3413/nukmed-00328-10-07
Intraoperative Sonography: A Technique for Localizing Focal Forms of Congenital Hyperinsulinism in the Pancreas
von Rohden, L.; Mohnike, K.; Mau, H.; Eberhard, T.; Mohnike, W.; et al. (10 authors)
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Ultraschall in der Medizin 32(2011), 74-80
DOI: 10.1055/s-0029-1245598
A 18F-labeled Fluorobutyl-substituted spirocyclic piperidine derivative as a selective radioligand for PET imaging of sigma1 receptors
Maisonial, A.; Große Maestrup, E.; Fischer, S.; Hiller, A.; Scheunemann, M.; et al. (11 authors)
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ChemMedChem 6(2011), 1401-1410
DOI: 10.1002/cmdc.201100108
A Novel Tetrabranched Neurotensin(8-13) Cyclam Derivative: Synthesis, 64Cu-Labeling and Biological Evaluation
Röhrich, A.; Bergmann, R.; Kretzschmann, A.; Noll, S.; Steinbach, J.; et al. (7 authors)
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Journal of Inorganic Biochemistry 105(2011), 821-832
DOI: 10.1016/j.jinorgbio.2011.02.011
Nanomaterials: applications in cancer imaging and therapy
Barreto, J. A.; O'Malley, W.; Kubeil, M.; Graham, B.; Stephan, H.; et al. (6 authors)
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Advanced Materials 23(2011)12, H18-H40
DOI: 10.1002/adma.201190041
Synthesis, structure determination and (radio-) fluorination of novel functionalized phosphanes suitable for the traceless Staudinger ligation
Mamat, C.; Franke, M.; Peppel, T.; Köckerling, M.; Steinbach, J.
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Tetrahedron 67(2011), 4521-4529
DOI: 10.1016/j.tet.2011.04.091
Synthesis and biological evaluation of new [Tc(N)(PS)]-based mixed-ligand compounds useful in design of target-specific radiopharmaceuticas: the 2-methoxyphenylpiperazine dithiocarbamate derivatives as example
Bolzati, C.; Salvarese, N.; Carta, D.; Refosco, F.; Dolmella, A.; et al. (8 authors)
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Journal of Biological Inorganic Chemistry 16(2011), 137-155
DOI: 10.1007/s00775-010-0712-4
[18F]1-(3-fluoropropyl)piperazines as model compounds for the radiofluorination of pyrido[2,3-d]pyrimidines
Grosse-Gehling, P.; Wuest, F. R.; Peppel, T.; Köckerling, M.; Mamat, C.
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Radiochimica Acta 99(2011), 365-373
DOI: 10.1524/ract.2011.1834
Synthesis and biological evaluation of novel 4-benzylpiperazine ligands for sigma-1 receptor imaging
Li, Z.-J.; Ren, H.-Y.; Cui, M.-C.; Deuther-Conrad, W.; Tang, R.-K.; et al. (9 authors)
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Bioorganic & Medicinal Chemistry 19(2011)9, 2911-2917
DOI: 10.1016/j.bmc.2011.03.037
Cross-Coupling Reactions as Valuable Tool for the Preparation of PET Radiotracers
Pretze, M.; Große-Gehling, P.; Mamat, C.
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Molecules 16(2011), 1129-1165
DOI: 10.3390/molecules16021129
In vitro binding profile and radiosynthesis of a novel 18F-labeled azaspirovesamicol analog as potential ligand for imaging of the vesicular acetylcholine transporter
Wenzel, B.; Hiller, A.; Fischer, S.; Sorger, D.; Deuther-Conrad, W.; et al. (9 authors)
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Journal of Labelled Compounds and Radiopharmaceuticals 54(2011), 426-432
DOI: 10.1002/jlcr.1891
High regiocontrol in the nucleophilic ring opening of 1-aralkyl-3,4-epoxypiperidines with amines – A short-step synthesis of 4-fluorobenzyltrozamicol and novel anilidopiperidines
Scheunemann, M.; Hennig, L.; Funke, U.; Steinbach, J.
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Tetrahedron 67(2011), 3448-3456
DOI: 10.1016/j.tet.2011.03.045
Assessment of alpha 7 nicotinic acetylcholine receptor availability in juvenile pig brain with [18F]NS10743
Deuther-Conrad, W.; Fischer, S.; Hiller, A.; Becker, G.; Cumming, P.; et al. (10 authors)
- European Journal of Nuclear Medicine and Molecular Imaging 38(2011)8, 1541-1549
Automated radiosynthesis of the thiol-reactive labeling agent N-[6-(4-[18F]fluorobenzylidene)aminooxyhexyl]maleimide ([18F]FBAM)
Knieß, T.; Kuchar, M.; Pietzsch, J.
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Applied Radiation and Isotopes 69(2011), 1226-1230
DOI: 10.1016/j.apradiso.2011.03.043
Synthesis, pharmacological activity and structure affinity relationships of spirocyclic σ1 receptor ligands with a (2-fluoroethyl) residue in 3-position
Große Maestrup, E.; Wiese, C.; Schepmann, D.; Brust, P.; Wünsch, B.
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Bioorganic & Medicinal Chemistry 19(2011), 393-405
DOI: 10.1016/j.bmc.2010.11.013
The serotonin transporter availability in untreated early-onset and late-onset patients with obsessive-compulsive disorder
Hesse, S.; Stengler, K.; Regenthal, R.; Patt, M.; Becker, G.-A.; et al. (15 authors)
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International Journal of Neuropsychopharmacology 14(2011), 1-12
DOI: 10.1017/S1461145710001604
Molecular imaging of σ receptors: synthesis and evaluation of the potent σ1 selective radioligand [18F]fluspidine
Fischer, S.; Wiese, C.; Grosse Maestrup, E.; Hiller, A.; Deuther-Conrad, W.; et al. (10 authors)
- European Journal of Nuclear Medicine and Molecular Imaging 38(2011)3, 540-551
Traumatic Brain Injury Elicits Similar Alterations in α7 Nicotinic Receptor Density in Two Different Experimental Models
Hoffmeister, P.-G.; Donat, C. K.; Schuhmann, M. U.; Voigt, C.; Walter, B.; et al. (9 authors)
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Neuromolecular Medicine 13(2011)1, 44-53
DOI: 10.1007/s12017-010-8136-4
ISSN: 1535-1084
Enantioselective σ1 receptor binding and biotransformation of the spirocyclic PET tracer 1’-Benzyl-3-(3-fluoropropyl)-3H-spiro[[2]benzofuran-1,4’-piperidine]
Wiese, C.; Große Maestrup, E.; Schepmann, D.; Grimme, S.; Humpf, H.-U.; et al. (7 authors)
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Chirality 23(2011), 148-154
DOI: 10.1002/chir.20893
Design, Synthesis and Preliminary in vitro and in vivo Pharmacological Evaluation of 2-{4-[4-(2,5-disubstituted thiazolyl)phenylethyl] piperazin-1-yl}-1,8-naphthyridine-3- carbonitriles as Atypical Antipsychotic Agents
Chandra Sekhar, K. V. G.; Rao, V. S.; Deuther-Conrad, W.; Reddy, A. S.; Brust, P.; et al. (6 authors)
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Journal of Enzyme Inhibition And Medicinal Chemistry 26(2011)4, 561-568
DOI: 10.3109/14756366.2010.537658
Implementation of 89Zr production and in vivo imaging of B-cells in mice with 89Zr-labeled anti B-cell antibodies by small animal PET/CT
Walther, M.; Gebhardt, P.; Grosse-Gehling, P.; Würbach, L.; Irmler, I.; et al. (11 authors)
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Applied Radiation and Isotopes 69(2011), 852-857
DOI: 10.1016/j.apradiso.2011.02.040